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author:

洪芳 (洪芳.) [1] | 胡建达 (胡建达.) [2] | 王文峰 (王文峰.) [3]

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CQVIP

Abstract:

通过大黄素的3位烷基化,1位保护及与叔胺反应实现了对大黄素的化学修饰。目标产物是一个季铵盐。测试了目标产物对白血病细胞Molt-4和人淋巴瘤细胞CA46的抗癌活性。结果表明目标产物的抗癌活性比大黄素约高10倍。

Keyword:

大黄素 季铵盐 抗白血病

Community:

  • [ 1 ] 福州大学化学化工学院,福州350108
  • [ 2 ] 福建医科大学附属协和医院,福州350001

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Source :

海峡药学

ISSN: 1006-3765

Year: 2012

Issue: 9

Volume: 24

Page: 254-256

Cited Count:

WoS CC Cited Count:

SCOPUS Cited Count:

ESI Highly Cited Papers on the List: 0 Unfold All

WanFang Cited Count:

Chinese Cited Count: -1

30 Days PV: 2

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