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Inventor:

薛金萍 (薛金萍.) [1] (Scholars:薛金萍) | 张凤玲 (张凤玲.) [2] | 黄琪 (黄琪.) [3] | 李俊 (李俊.) [4]

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incoPat

Abstract:

本发明公开了一种分子靶向抗癌光敏剂埃罗替尼 酞菁轭合物及其应用,在金属酞菁大环周边引入带有烷氧长链的埃罗替尼结构单元,可以增加其两亲性、生物相容性、光敏剂的靶向性。该轭合物不容易聚集,有利于提高细胞摄取率;同时该类化合物结构单一,不存在异构体,产品容易提纯。该化合物有望提高光动力治疗中光敏剂的靶向性,同时增强光动力治疗中光敏剂的活性。本发明合成方法比较简单,副反应少,产率较高,原料易得,成本低,有利于工业化生产。

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Patent Info :

Type: 发明授权

Patent No.: CN201410791090.0

Filing Date: 2013/6/18

Publication Date: 2016/10/26

Pub. No.: CN104447769B

公开国别: CN

Applicants: 福州大学

Legal Status: 授权

Cited Count:

WoS CC Cited Count:

SCOPUS Cited Count:

ESI Highly Cited Papers on the List: 0 Unfold All

WanFang Cited Count:

Chinese Cited Count:

30 Days PV: 4

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