3-Aminoindole Synthesis from 2-Nitrochalcones and Ammonia or Primary Amines - Details

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Abstract：

A　step-economic　strategy　for　3-aminoindoles　synthesis　with　ammonia　or　primary　amines　as　“N”　source　under　transition-metal-free　conditions　was　achieved.　A　series　of　3-aminoindoles　was　obtained　with　abundant　“N”　source　featuring　high　efficiency,　mild　conditions,　environmental　friendliness　and　scalability.　Efficient　syntheses　of　the　intermediates　of　COX-2　inhibitor　and　tubulin　polymerization　inhibitor　were　successfully　accomplished　with　this　newly　developed　strategy.　(Figure　presented.).　©　2019　Wiley-VCH　Verlag　GmbH　&　Co.　KGaA,　Weinheim

Keyword：

2-nitrochalcone; 3-aminoindole; ammonia; metal-free; primary amines

Community：

[ 1 ] [Zhang, G.]Institute of Next Generation Matter Transformation, College of Material Sciences Engineering at, Huaqiao University, 668 Jimei Boulevard, Xiamen, Fujian 361021, China
[ 2 ] [Lin, L.]College of Chemistry and Chemical Engineering, Xiamen University, Xiamen, 361005, China
[ 3 ] [Yang, K.]College of Chemistry, Fuzhou University, Fuzhou, 350116, China
[ 4 ] [Wang, S.]Institute of Next Generation Matter Transformation, College of Material Sciences Engineering at, Huaqiao University, 668 Jimei Boulevard, Xiamen, Fujian 361021, China
[ 5 ] [Feng, Q.]Institute of Next Generation Matter Transformation, College of Material Sciences Engineering at, Huaqiao University, 668 Jimei Boulevard, Xiamen, Fujian 361021, China
[ 6 ] [Zhu, J.]College of Chemistry and Chemical Engineering, Xiamen University, Xiamen, 361005, China
[ 7 ] [Song, Q.]Institute of Next Generation Matter Transformation, College of Material Sciences Engineering at, Huaqiao University, 668 Jimei Boulevard, Xiamen, Fujian 361021, China
[ 8 ] [Song, Q.]College of Chemistry, Fuzhou University, Fuzhou, 350116, China

Reprint 's Address：

[Zhu, J.]College of Chemistry and Chemical Engineering, Xiamen UniversityChina

Email：

jun.zhu@xmu.edu.cn

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Source ：

Advanced Synthesis and Catalysis

ISSN： 1615-4150

Year： 2019

Issue： 16

Volume： 361

Page： 3718-3722

5 . 8 5 1

JCR@2019

4 . 4 0 0

JCR@2023

ESI HC Threshold：184

JCR Journal Grade：1

CAS Journal Grade：1

Cited Count：

WoS CC Cited Count：

SCOPUS Cited Count： 14

ESI Highly Cited Papers on the List： 0 Unfold All

WanFang Cited Count：

Chinese Cited Count：

30 Days PV： 4

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